Method Development in the Pharmaceutical Field

The purpose of method development is to establishensures the samples are sufficiently clean and
the applicability of an analytical method for itstherefore able to maintain the shelf-life of the
intended use on a certain sample. There are manyanalytical instrument used. If unsatisfactory results
tests that need to be carried out in theare obtained, some adjustment has to be made to
pharmaceutical field, such as assay, dissolution,the method. For example, for a method developed
identification and related substance. Each of theseusing high performance liquid chromatography (HPLC),
tests, particularly the quantitative analysis has to beadjustment can be made to various stages of the
developed for its fit for use before approving it foranalysis such as sample preparation, mobile phase and
routine application.the stationary phase. The extensiveness of the
How to go about developing a method? Usually themethod development work depends on the
first step is literature search. This step includes thecomplexity of the sample as well as the instrument
reviewing of analytical methods from monographs,used.
scientific journals, drug suppliers and analyticalAfter development stage, the method has to be
instrument companies. For some drugs, the contentvalidated for the parameters below:
can be analyzed employing various methods, for• Linearity refers to the relationship between the
instance, high performance liquid chromatographytest results and the concentration of the drug
(HPLC), ultra-violet spectrophotometer and titration.analyzed
Therefore, it is important to review the available• Range is the maximum and minimum
methods according to its application. Examples ofconcentration levels that have been proven to have
parameters in a method that can be evaluated are itsaccuracy, precision and linearity
sensitivity, specificity and available resources. Usually• Accuracy measures the closeness of the test
for a pharmaceutical manufacturing company,results to the true value
methods from monographs are preferred due to its• Precision is related to both the instrument and
validity. However, recently, the requirement tomethod. This parameter measures the closeness of
validate monograph methods is increasing.the test results to each other
After selecting the most suitable method, the• Specificity refers to the ability of the method to
laboratory personnel need to try out the method.separate the analyte from other ingredients present
During this phase, applicability of the method in termsin the sample
of sample preparation and analytical instrument set up• Sensitivity is the parameter pertaining to the
is evaluated. Sample preparation is important toability of the method to quantify and detect the
ensure accurate and reproducible results. It alsolowest amount of the analyte.